Bioheterocycles 2019

XVIII International Conference on Heterocycles in Bioorganic Chemistry

 Ghent, Belgium    June 17-20, 2019

Plenary lectures

Heterocyclic Chemistry in Drug Development (PL07)

Prof. Wim DE BORGGRAEVE
Prof. Wim DE BORGGRAEVE
KULEUVEN, Heverlee, Belgium
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Heterocycles To Control Immune Cell Function (PL03)

Prof. David FAIRLIE
Prof. David FAIRLIE
UNIVERSITY OF QUEENSLAND, Brisbane, Australia
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Multiple Conjugation Reactions on Peptides and Oligonucleotides (PL06)

Prof. Anna GRANDAS
Prof. Anna GRANDAS
UNIVERSITY OF BARCELONA, Barcelona, Spain
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Synthesis of Heterocyles Using Visible Light Photocatalysis (PL04)

Prof. Burkhard KÖNIG
Prof. Burkhard KÖNIG
UNIVERSITY OF REGENSBURG, Regensburg, Germany
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The Beautiful Simplicity of Rearrangements (PL05)

Prof. Nuno MAULIDE
Prof. Nuno MAULIDE
UNIVERSITY OF VIENNA, Vienna, Austria
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Heterocycles as Key Features of New Starting Points for Drug Discovery (PL01)

Dr Peter MEIER
Dr Peter MEIER
NOVARTIS PHARMA AG, Basel, Switzerland
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A Journey in Heteroaromatic Scaffolds as Protein Kinase Inhibitors (PL02)

Prof. Pascale MOREAU
Prof. Pascale MOREAU
UNIVERSITY OF CLERMONT AUVERGNE, Aubičre, France
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Invited lectures

Bacterial Quinolones and Derivatives: New Drugs for Bad Bugs (IL03)

Dr Thomas BOTTCHER
Dr Thomas BOTTCHER
UNIVERSITY OF KONSTANZ, Konstanz, Germany
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Heterocycles as a Route to New Chemical Space for Drug Discovery (IL09)

Prof. James BULL
Prof. James BULL
IMPERIAL COLLEGE, London, United Kingdom
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Heterocycles and Neglected Diseases: Still a Role for Total Synthesis (IL08)

Prof. Adrian DOBBS
Prof. Adrian DOBBS
UNIVERSITY OF GREENWICH, Kent, United Kingdom
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Development of Enzyme Inhibitors and Multi-target-directed Ligands for Treating Neurodegenerative Diseases (IL01)

Prof. Stanislav GOBEC
Prof. Stanislav GOBEC
UNIVERSITY OF LJUBLJANA, Ljubljana, Slovenia
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Vitamin B12 – an Intriguing Bioheterocycle (IL04)

Prof. Dorota GRYKO
Prof. Dorota GRYKO
INSTITUTE OF ORGANIC CHEMISTRY PAS, Warsaw, Poland
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A journey with Saponins (IL07)

Dr Martina LAHMANN
Dr Martina LAHMANN
BANGOR UNIVERSITY, Wales, United Kingdom
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Functionalization of Aromatic Heterocycles Using Bases Derived from LiTMP (IL05)

Prof. Florence MONGIN
Prof. Florence MONGIN
UNIVERSITY OF RENNES, Rennes, France
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Leveraging Carbonylation and N-acyl imine Chemistry in Heterocycle Synthesis (IL06)

Dr Luke ODELL
Dr Luke ODELL
UNIVERSITY OF UPPSALA, Uppsala, Sweden
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Biologically Active Azaheterocycles Containing a Ferrocene Moiety (IL10)

Prof. Niko S. RADULOVIC
Prof. Niko S. RADULOVIC
UNIVERSITY OF NIS, Nis, Serbia

Expanding the Chemical Space of Chiral Trifunctional Building Blocks by Stereoselective Synthesis from Natural Terpenes (IL02)

Prof. Zsolt SZAKONYI
Prof. Zsolt SZAKONYI
UNIVERSITY OF SZEGED, Szeged, Hungary
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Oral Communications

Chiral Piperidines from Pyridines: the Meta-Substitution Challenge in Asymmetric Hydrogenation (OC02)

Dr Paul ALSTERS
Dr Paul ALSTERS
INNOSYN B.V., Geleen, The Netherlands
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Silil-Prins Cyclization: Towards the Synthesis of Medium Sized Heterocycles (OC01)

Prof. Asuncion BARBERO
Prof. Asuncion BARBERO
UNIVERSITY OF VALLADOLID, Valladolid, Spain

Combining Isocyanides with Carbon Dioxide for Heterocycle Synthesis (OC20)

Mr Jeroen BOMON
Mr Jeroen BOMON
UNIVERSITEIT ANTWERPEN, Antwerpen, Belgium
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Towards DNA-Encoded Heterocycle Libraries - DNA-Compatible Povarov and Groebke Reactions by Micellar Broensted Acid Catalysis (OC24)

Dr Andreas BRUNSCHWEIGER
Dr Andreas BRUNSCHWEIGER
TU DORTMUND, Dortmund, Germany
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The Phenanthridine PJ-34 Exclusively Eradicates Human cancer Cells (OC16)

Prof. Malka COHEN-ARMON
Prof. Malka COHEN-ARMON
TEL-AVIV UNIVERSITY, Tel-Aviv, Israel
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Hydrogen Peroxide and Hydrohalic Acid-Mediated Synthesis of Ring-Fused Benzimidazolequinone Anti-Cancer Agents (OC03)

Mr Darren CONBOY
Mr Darren CONBOY
KINGSTON UNIVERSITY LONDON, Kingston upon Thames, United Kingdom
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First Solid-Phase Strategy for the Total Synthesis of Fengycin Derivatives, a Class of Cyclic Lipodepsipeptides (OC05)

Dr Lidia FELIU
Dr Lidia FELIU
LIPPSO, UNIVERSITY OF GIRONA, Girona, Spain
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Regioselective C-H Arylation of Nitro Heterocycles and Further Transformation of Manipulable Nitro Group (OC23)

Dr Viktor IAROSHENKO
Dr Viktor IAROSHENKO
POLISH ACADEMY OF SCIENCES, Lodz, Poland
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Thionations Using a P4S10-Pyridine Complex (OC04)

Ms Ngarita KINGI
Ms Ngarita KINGI
VIRONOVA MEDICAL AB, Stockholm, Sweden
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'Stretched' Analogs of Piperidine, Piperazine, and Morpholine: Advanced Building Blocks for Drug Discovery (OC18)

Dr Ivan KONDRATOV
Dr Ivan KONDRATOV
ENAMINE, Kiev, Ukraine
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Structurally Simple Cytosine Peptidomimetics as Potent Cardioprotectors in Myocardial Ischemia (MI) Mouse Model: Design, Synthesis And Biological Evaluation (OC12)

Dr Edward KORSHIN
Dr Edward KORSHIN
BAR-ILAN UNIVERSITY, Ramat Gan, Israel
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Playing with Properties of Biologically Active Compounds: High-Throughput Conjugation of Drug-Like Molecules for Chemical Biology (OC22)

Ms Sona KRAJCOVICOVA
Ms Sona KRAJCOVICOVA
PALACKY UNIVERSITY, Olomouc, Czech Republic
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Biradical Formation by Deprotonation in Conjugated 2-Amino/Imino Thiazole Derivatives (OC13)

Prof. Francisco LOPEZ-CALAHORRA
Prof. Francisco LOPEZ-CALAHORRA
UNIVERSITAT DE BARCELONA, Barcelona, Spain
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Application of Tsunoda reagent to the convenient synthesis of drug-like pyrazoles (OC15)

Dr Olivier LORTHIOIR
Dr Olivier LORTHIOIR
ASTRAZENECA, Cambridge, United Kingdom

The Magic of Wood and Light – New Concepts for Synthetic Chemistry (OC10)

Prof. Till OPATZ
Prof. Till OPATZ
JOHANNES GUTENBERG-UNIVERSITY, Mainz, Germany

Hydroxylated Heterocycles as a Bioisosteric Tool to Modulate the Carboxylic Function (OC08)

Dr Agnese Chiara PIPPIONE
Dr Agnese Chiara PIPPIONE
UNIVERSITY OF TURIN, Torino, Italy
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Kolbe Anodic Decarboxylation as a Green Way to Access Pyrrolidinones (OC21)

Ms Mathilde QUERTENMONT
Ms Mathilde QUERTENMONT
UNIVERSITÉ CATHOLIQUE DE LOUVAIN, La Hulpe, Belgium
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Tweaking the Blebbistatin Scaffold Towards Better Pharmacological Tools (OC09)

Dr Bart ROMAN
Dr Bart ROMAN
GHENT UNIVERSITY, Ghent, Belgium

Synthesis and in vitro -Glucosidase Inhibitory Activity of Polyhydroxylated 2-Styrylchromones (OC17)

Dr Clementina SANTOS
Dr Clementina SANTOS
INSTITUTO POLITÉCNICO DE BRAGANÇA, Braganca, Portugal
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Small but Selective: Developing Chemical Probes for PKN/PRK2 (OC14)

Ms Fiona SCOTT
Ms Fiona SCOTT
SUSSEX DRUG DISCOVERY CENTRE, Falmer, United Kingdom
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Biologically Active Oxygen and Nitrogen Heterocyclic Compounds from Cycloaddition and Conjugate Addition Reactions On Chromones (OC19)

Prof. Artur M.S. SILVA
Prof. Artur M.S. SILVA
UNIVERSITY OF AVEIRO, Aveiro, Portugal
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Synthesis of Enantioenriched 3-Isobenzofuranones Using Chiral Organomagnesiates (OC11)

Dr Sabrina TOUCHET
Dr Sabrina TOUCHET
UNIVERSITÉ DE LORRAINE, Vandoeuvre-les-Nancy, France
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Design and Synthesis of New Nitrogen-Containing Heterocycles for the Treatment of Mechanical Allodynia (OC06)

Ms Alexia VISSEQ
Ms Alexia VISSEQ
INSTITUT DE CHIMIE DE CLERMONT FERRAND, AUBIERE, France
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